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Nagavarakishore Pillarsetty Selected Research

6- amino- 8- ((6- iodo- 1,3- benzodioxol- 5- yl)thio)- N- (1- methylethyl)- 9H-purine-9-propanamine

10/2020First-in-Human Trial of Epichaperome-Targeted PET in Patients with Cancer.
1/2020Measuring Tumor Epichaperome Expression Using [124I] PU-H71 Positron Emission Tomography as a Biomarker of Response for PU-H71 Plus Nab-Paclitaxel in HER2-Negative Metastatic Breast Cancer.
9/2011Affinity-based proteomics reveal cancer-specific networks coordinated by Hsp90.

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Nagavarakishore Pillarsetty Research Topics

Disease

34Neoplasms (Cancer)
01/2022 - 01/2003
3Glioblastoma (Glioblastoma Multiforme)
01/2022 - 12/2012
3Prostatic Neoplasms (Prostate Cancer)
01/2022 - 10/2009
3Pancreatic Neoplasms (Pancreatic Cancer)
01/2022 - 12/2017
2Adenocarcinoma
10/2021 - 01/2020
2Breast Neoplasms (Breast Cancer)
01/2020 - 08/2009
2BCR-ABL Positive Chronic Myelogenous Leukemia (Chronic Myelogenous Leukemia)
09/2011 - 01/2010
2Carcinoma (Carcinomatosis)
07/2008 - 01/2003
1Small Cell Lung Carcinoma (Small Cell Lung Cancer)
01/2022
1Purpura
01/2022
1Alzheimer Disease (Alzheimer's Disease)
01/2021
1COVID-19
01/2021
1Anaplastic Thyroid Carcinoma
12/2020
1Melanoma (Melanoma, Malignant)
12/2020
1Fever (Fevers)
01/2020
1Thyroid Neoplasms (Thyroid Cancer)
11/2016
1Sarcoma (Soft Tissue Sarcoma)
05/2014
1Gastrointestinal Stromal Tumors (Gastrointestinal Stromal Tumor)
05/2014
1Fibrosis (Cirrhosis)
05/2014
1Glioma (Gliomas)
12/2012
1Brain Neoplasms (Brain Tumor)
12/2012
1Neoplasm Metastasis (Metastasis)
08/2009
1Lymphoma (Lymphomas)
01/2003

Drug/Important Bio-Agent (IBA)

7Pharmaceutical PreparationsIBA
01/2022 - 12/2012
4GemcitabineFDA Link
01/2022 - 12/2017
4LigandsIBA
01/2022 - 07/2011
36- amino- 8- ((6- iodo- 1,3- benzodioxol- 5- yl)thio)- N- (1- methylethyl)- 9H-purine-9-propanamineIBA
10/2020 - 09/2011
3Biomarkers (Surrogate Marker)IBA
09/2020 - 12/2015
3Phosphotransferases (Kinase)IBA
02/2011 - 11/2007
2Capecitabine (Xeloda)FDA Link
01/2022 - 01/2020
2Mitogen-Activated Protein Kinase Kinases (MEKs)IBA
10/2021 - 12/2020
2ProteomeIBA
01/2021 - 09/2011
2Proteins (Proteins, Gene)FDA Link
01/2021 - 09/2011
2Liposomes (Liposome)IBA
11/2013 - 02/2011
2Dasatinib (BMS 354825)FDA Link
12/2012 - 02/2012
2AndrogensIBA
10/2009 - 01/2003
22'-fluoro-5-ethylarabinosyluracil (FEAU)IBA
08/2009 - 04/2008
2LuciferasesIBA
08/2009 - 07/2008
1Indicators and Reagents (Reagents)IBA
01/2022
11,4,7- triazacyclononane- N,N',N''- triacetic acid (NOTA)IBA
01/2022
1N- (2- amino- 3- (4- isothiocyanatophenyl)propyl)cyclohexane- 1,2- diamine- N,N',N',N'',N''- pentaacetic acidIBA
01/2022
1Pentetic Acid (DTPA)FDA LinkGeneric
01/2022
1Androgen Receptors (Androgen Receptor)IBA
01/2022
1Immune Checkpoint InhibitorsIBA
10/2021
11- (2'- deoxy- 2'- fluoro- arabinofuranosyl)cytosineIBA
01/2021
1PEGPH20IBA
01/2021
1Hyaluronoglucosaminidase (Hyaluronidase)FDA Link
01/2021
1AntibodiesIBA
01/2021
1Mitogen-Activated Protein KinasesIBA
12/2020
1trametinibIBA
12/2020
1Extracellular Signal-Regulated MAP Kinases (Extracellular Signal Regulated Kinases)IBA
12/2020
1N 30IBA
10/2020
1Fluorouracil (Carac)FDA LinkGeneric
01/2020
1130-nm albumin-bound paclitaxelIBA
01/2020
1Adenosine Triphosphate (ATP)IBA
01/2020
1CytosineIBA
12/2017
1IodidesIBA
11/2016
1Poly(ADP-ribose) Polymerases (Poly ADP Ribose Polymerase)IBA
12/2015
1pexidartinibIBA
05/2014
1Imatinib Mesylate (Gleevec)FDA Link
05/2014
1Peptides (Polypeptides)IBA
11/2013
1CyclooctanesIBA
11/2013
1ProdrugsIBA
04/2013
1EnzymesIBA
04/2013
1Laminin ReceptorsIBA
04/2013
1MicellesIBA
12/2012
1Proto-Oncogene Proteins c-sis (Platelet Derived Growth Factor B)IBA
12/2012
1FluorineIBA
12/2012
1Platelet-Derived Growth Factor Receptors (Platelet-Derived Growth Factor Receptor)IBA
12/2012
1Biological ProductsIBA
12/2012
1Oncogene Proteins (Oncogene Protein)IBA
09/2011
1LipidsIBA
02/2011
1ErbB Receptors (EGF Receptor)IBA
02/2011
12- (4- iodophenylamino)pyrido(2,3- d)pyrimidin- 7- oneIBA
01/2010
12-18F-fluoropropionic acidIBA
10/2009
1AcidsIBA
10/2009
1Firefly LuciferasesIBA
08/2009
1Transforming Growth Factor beta (TGF-beta)IBA
08/2009
1AntigensIBA
07/2008
1Renilla LuciferasesIBA
07/2008
1GuanineIBA
05/2008
12'- fluoro- 2'- deoxy- 5- fluoroethyl- 1- beta- D- arabinofuranosyl uracilIBA
04/2008
1Tyrosine (L-Tyrosine)FDA Link
11/2007
1GoldIBA
01/2003
1tetrakis((trishydroxymethyl)phosphine)gold(I)IBA
01/2003

Therapy/Procedure

13Therapeutics
01/2022 - 07/2008
2Radioimmunotherapy
01/2022 - 01/2022
1Castration
01/2022
1Euthanasia (Mercy Killing)
01/2022
1Injections
01/2021
1Precision Medicine
11/2019
1Molecular Targeted Therapy
05/2014
1Aftercare (After-Treatment)
01/2010